Browsing Faculty of Health Sciences by Author "Parapini, Silvia"
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Facile preparation of N-glycosylated 10-piperazinyl artemisinin derivatives and evaluation of their antimalarial and cytotoxic activities
Wu, Yuet; Wong, Ho Ning; Haynes, Richard K.; Parapini, Silvia; Williams, Ian D. (MDPI, 2018)According to the precepts that C-10 amino-artemisinins display optimum biological activities for the artemisinin drug class, and that attachment of a sugar enhances specificity of drug delivery, polarity and solubility so ... -
Inhibition of metalloproteinase-9 secretion and gene expression by artemisinin derivatives
Magenta, Daniele; Haynes, Richard K.; Sangiovanni, Enrico; Basilico, Nicoletta; Parapini, Silvia (Elsevier, 2014)Malaria remains one of the world's most common infectious diseases, being responsible for more deaths than any other communicable disease except tuberculosis. There is strong evidence that tumour necrosis factor α and ...